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AAK1 inhibitor 25A
CAS No. ——
AAK1 inhibitor 25A( —— )
Catalog No. M16970 CAS No. ——
AAK1 inhibitor 25A is a potent, selective inhibitor of AAK1 and the closely related kinase BMP2K with Ki of 8 nM (AAK1).
Purity : >98% (HPLC)
COA
Datasheet
HNMR
HPLC
MSDS
Handing Instructions
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Biological Information
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Product NameAAK1 inhibitor 25A
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NoteResearch use only, not for human use.
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Brief DescriptionAAK1 inhibitor 25A is a potent, selective inhibitor of AAK1 and the closely related kinase BMP2K with Ki of 8 nM (AAK1).
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DescriptionAAK1 inhibitor 25A is a potent, selective inhibitor of AAK1 and the closely related kinase BMP2K with Ki of 8 nM (AAK1); displays selectivity over the other members of the subfamily, Numb-associated kinases GAK and STK16, in a TR-FRET binding displacement assay; binds to BMP2K in live HEK293T cells with an IC50 of 602 nM.
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In Vitro——
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In Vivo——
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Synonyms——
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PathwayOthers
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TargetAAK1
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RecptorAAK1
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Research Area——
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Indication——
Chemical Information
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CAS Number——
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Formula Weight396.465
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Molecular FormulaC20H20N4O3S
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Purity>98% (HPLC)
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Solubility——
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SMILES——
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Chemical NameN-(6-(3-(cyclopropanesulfonamido)phenyl)-1H-indazol-3-yl)cyclopropanecarboxamide
Shipping & Storage Information
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Storage(-20℃)
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ShippingWith Ice Pack
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Stability≥ 2 years
Reference
1. Agajanian MJ, et al. Cell Rep. 2019 Jan 2;26(1):79-93.e8.
molnova catalog
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